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Critical Reviews™ in Therapeutic Drug Carrier Systems

Publication de 6  numéros par an

ISSN Imprimer: 0743-4863

ISSN En ligne: 2162-660X

The Impact Factor measures the average number of citations received in a particular year by papers published in the journal during the two preceding years. 2017 Journal Citation Reports (Clarivate Analytics, 2018) IF: 2.7 To calculate the five year Impact Factor, citations are counted in 2017 to the previous five years and divided by the source items published in the previous five years. 2017 Journal Citation Reports (Clarivate Analytics, 2018) 5-Year IF: 3.6 The Immediacy Index is the average number of times an article is cited in the year it is published. The journal Immediacy Index indicates how quickly articles in a journal are cited. Immediacy Index: 0.8 The Eigenfactor score, developed by Jevin West and Carl Bergstrom at the University of Washington, is a rating of the total importance of a scientific journal. Journals are rated according to the number of incoming citations, with citations from highly ranked journals weighted to make a larger contribution to the eigenfactor than those from poorly ranked journals. Eigenfactor: 0.00023 The Journal Citation Indicator (JCI) is a single measurement of the field-normalized citation impact of journals in the Web of Science Core Collection across disciplines. The key words here are that the metric is normalized and cross-disciplinary. JCI: 0.39 SJR: 0.42 SNIP: 0.89 CiteScore™:: 5.5 H-Index: 79

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Pharmacodynamic Aspects of Modes of Drug Administration for Optimization of Drug Therapy

Volume 16, Numéro 6, 1999, 70 pages
DOI: 10.1615/CritRevTherDrugCarrierSyst.v16.i6.20
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RÉSUMÉ

Because of various pharmacodynamic properties, such as the nonlinearity of the concentration-effect relationship, activation of feedback homeostatic mechanisms, induction of pharmacodynamic tolerance, etc., administration of die same dose of drug by different modes is expected to produce different outcomes. This review clarifies the theoretical and practical aspects of the impact of different modes of drag administration on the magnitude of response, and hence on therapy outcomes. It discusses how the interrelationship between the pharmacodynamic properties and die drug input function affects die magnitude of response. To demonstrate this special dimension of drug therapy, relevant pharmacodynamic data was obtained for drugs with different therapeutic applications, including antibiotics, analgesics, diuretics, anti-cancer, anti-ulcer, anti-inflammatory, anti-hypertensive, lipid-lowering anti-parkinsonian, and immunosuppressive drugs. These examples provide guidelines for implementing the role of the mode of drug administration (including rate, schedule, and route of drug treatment) during drug development or optimization of drug therapy.

CITÉ PAR
  1. Stepensky David, The Øie–Tozer model of drug distribution and its suitability for drugs with different pharmacokinetic behavior, Expert Opinion on Drug Metabolism & Toxicology, 7, 10, 2011. Crossref

  2. Bomma Ramesh, Veerabrahma Kishan, Development of gastroretentive drug delivery system for cefuroxime axetil:In vitroandin vivoevaluation in human volunteers, Pharmaceutical Development and Technology, 18, 5, 2013. Crossref

  3. Gaur Praveen Kumar, Mishra Shikha, Kumar Avdhesh, Panda Bibhu Prasad, Development and optimization of gastroretentive mucoadhesive microspheres of gabapentin by Box–Behnken design, Artificial Cells, Nanomedicine, and Biotechnology, 42, 3, 2014. Crossref

  4. Klausner Eytan A., Lavy Eran, Stepensky David, Cserepes Eva, Barta Miklos, Friedman Michael, Hoffman Amnon, Furosemide Pharmacokinetics and Pharmacodynamics following Gastroretentive Dosage Form Administration to Healthy Volunteers, The Journal of Clinical Pharmacology, 43, 7, 2003. Crossref

  5. Rhee Yun-Seok, Park Seok, Lee Tae-Won, Park Chun-Woong, Nam Tae-Young, Oh Tack-Oon, Jeon Ji-Woong, Han Sang Beom, Lee Dong-Soo, Park Eun-Seok, In Vitro/in Vivo relationship of gabapentin from a sustained-release tablet formulation: A pharmacokinetic study in the beagle dog, Archives of Pharmacal Research, 31, 7, 2008. Crossref

  6. Barbanoj MJ, Ballester MR, Antonijoan RM, Puntes M, Gropper S, Santos B, Albet C, Guglietta A, A BIOAVAILABILITY/BIOEQUIVALENCE AND PHARMACOKINETIC STUDY OF TWO ORAL DOSES OF TORASEMIDE (5 AND 10 mg): PROLONGED-RELEASE VERSUS THE CONVENTIONAL FORMULATION, Clinical and Experimental Pharmacology and Physiology, 36, 5-6, 2009. Crossref

  7. Barbanoj M.J., Ballester M.R., Antonijoan R.M., Gich I., Pelagio P., Gropper S., Santos B., Guglietta A., Comparison of repeated-dose pharmacokinetics of prolonged-release and immediate-release torasemide formulations in healthy young volunteers, Fundamental & Clinical Pharmacology, 23, 1, 2009. Crossref

  8. Hoffman Amnon, Horwitz Ehud, Hess Shmuel, Cohen-Poradosu Ronit, Kleinberg Lilach, Edelberg Anna, Shapiro Mervyn, Implications on Emergence of Antimicrobial Resistance as a Critical Aspect in the Design of Oral Sustained Release Delivery Systems of Antimicrobials, Pharmaceutical Research, 25, 3, 2008. Crossref

  9. Klausner Eytan A, Lavy Eran, Friedman Michael, Hoffman Amnon, Expandable gastroretentive dosage forms, Journal of Controlled Release, 90, 2, 2003. Crossref

  10. Stepensky David, Friedman Michael, Srour Wassim, Raz Itamar, Hoffman Amnon, Preclinical evaluation of pharmacokinetic–pharmacodynamic rationale for oral CR metformin formulation, Journal of Controlled Release, 71, 1, 2001. Crossref

  11. Chavanpatil Mahesh, Jain Paras, Chaudhari Sachin, Shear Rajesh, Vavia Pradeep, Development of sustained release gastroretentive drug delivery system for ofloxacin: In vitro and in vivo evaluation, International Journal of Pharmaceutics, 304, 1-2, 2005. Crossref

  12. Mukker Jatinder Kaur, Singh Ravi Shankar Prasad, Derendorf Hartmut, Pharmacokinetic and pharmacodynamic implications in inhalable antimicrobial therapy, Advanced Drug Delivery Reviews, 85, 2015. Crossref

  13. Prinderre Pascal, Sauzet Christophe, Fuxen Claus, Advances in gastro retentive drug-delivery systems, Expert Opinion on Drug Delivery, 8, 9, 2011. Crossref

  14. Hu Liandong, Li Li, Yang Xun, Liu Wei, Yang Jianxue, Jia Yanhong, Shang Chuang, Xu Hongxin, Floating matrix dosage form for dextromethorphan hydrobromide based on gas forming technique: In vitro and in vivo evaluation in healthy volunteers, European Journal of Pharmaceutical Sciences, 42, 1-2, 2011. Crossref

  15. Stepensky David, Use of unbound volumes of drug distribution in pharmacokinetic calculations, European Journal of Pharmaceutical Sciences, 42, 1-2, 2011. Crossref

  16. Klausner Eytan A, Eyal Sara, Lavy Eran, Friedman Michael, Hoffman Amnon, Novel levodopa gastroretentive dosage form: in-vivo evaluation in dogs, Journal of Controlled Release, 88, 1, 2003. Crossref

  17. Hoffman Amnon, Stepensky David, Lavy Eran, Eyal Sara, Klausner Eytan, Friedman Michael, Pharmacokinetic and pharmacodynamic aspects of gastroretentive dosage forms, International Journal of Pharmaceutics, 277, 1-2, 2004. Crossref

  18. Goole J., Van Gansbeke B., Pilcer G., Deleuze Ph., Blocklet D., Goldman S., Pandolfo M., Vanderbist F., Amighi K., Pharmacoscintigraphic and pharmacokinetic evaluation on healthy human volunteers of sustained-release floating minitablets containing levodopa and carbidopa, International Journal of Pharmaceutics, 364, 1, 2008. Crossref

  19. Reich Reuven, Hoffman Amnon, Suresh R. Rama, Shai Ofra, Frant Julia, Maresca Alfonso, Supuran Claudiu T., Breuer Eli, Carbamoylphosphonates inhibit autotaxin and metastasis formationin vivo, Journal of Enzyme Inhibition and Medicinal Chemistry, 30, 5, 2015. Crossref

  20. Pillai Omathanu, Dhanikula Anand Babu, Panchagnula Ramesh, Drug delivery: an odyssey of 100 years, Current Opinion in Chemical Biology, 5, 4, 2001. Crossref

  21. Hoffman Amnon, Qadri Bashir A., Drug Delivery: Gastro-Retentive Systems, in Encyclopedia of Biomedical Polymers and Polymeric Biomaterials, 2016. Crossref

  22. Satapathy Trilochan, Panda Prasana K., Goyal Amit K., Rath Goutam, Evaluation of Anti-GERD Activity of Gastro Retentive Drug Delivery System of Itopride Hydrochloride, Artificial Cells, Blood Substitutes, and Biotechnology, 38, 4, 2010. Crossref

  23. Bélair Jacques, Rimbu Andreea, Time Delays in Drug Administration: Effect, Transit, Tricks and Oscillations∗∗Financial support of the Natural Sciences and Enginering Research Council (NSERC, Canada) [Discovery Grant to JB], the Fonds de Recherche du Québec –Nature et Technologies (FRQNT, Québec) [Team Grant to JB and Doctoral Fellowship to AR] and Université de Montréal is acknowledged., IFAC-PapersOnLine, 48, 12, 2015. Crossref

  24. Ashraf Muhammad Umer, Hussain Muhammad Ajaz, Bashir Sajid, Haseeb Muhammad Tahir, Hussain Zakir, Quince seed hydrogel (glucuronoxylan): Evaluation of stimuli responsive sustained release oral drug delivery system and biomedical properties, Journal of Drug Delivery Science and Technology, 45, 2018. Crossref

  25. Wu Benjamin, Sy Sherwin K. B., Derendorf Hartmut, Principles of Applied Pharmacokinetic–Pharmacodynamic Modeling, in Fundamentals of Antimicrobial Pharmacokinetics and Pharmacodynamics, 2014. Crossref

  26. Stepensky David, Kleinberg Lilach, Hoffman Amnon, Bone as an Effect Compartment, Clinical Pharmacokinetics, 42, 10, 2003. Crossref

  27. Stepensky David, Friedman Michael, Raz Itamar, Hoffman Amnon, Pharmacokinetic-Pharmacodynamic Analysis of the Glucose-Lowering Effect of Metformin in Diabetic Rats Reveals First-Pass Pharmacodynamic Effect, Drug Metabolism and Disposition, 30, 8, 2002. Crossref

  28. Sy Sherwin K. B., Derendorf Hartmut, Pharmacometrics in Bacterial Infections, in Applied Pharmacometrics, 14, 2014. Crossref

  29. Sheikh Fatima Akbar, Hussain Muhammad Ajaz, Ashraf Muhammad Umer, Haseeb Muhammad Tahir, Farid-ul-Haq Muhammad, Linseed hydrogel based floating drug delivery system for fluoroquinolone antibiotics: Design, in vitro drug release and in vivo real-time floating detection, Saudi Pharmaceutical Journal, 28, 5, 2020. Crossref

  30. Yamani Lamya, Alamri Aisha, Alsultan Afnan, Alfifi Somaya, Ansari Mohammad Azam, Alnimr Amani, Inverse correlation between biofilm production efficiency and antimicrobial resistance in clinical isolates of Pseudomonas aeruginosa, Microbial Pathogenesis, 157, 2021. Crossref

  31. Patil Mayuri B., Maru Avish D., Bhadane Jayshree S., Formulation and Evaluation of Sustained Release Bilayer Matrix Tablet of Glimepiride and Metformin Hydrochloride, Asian Journal of Research in Pharmaceutical Sciences, 2021. Crossref

  32. Shang Wenting, Peng Li, Guo Pengyu, Hui Hui, Yang Xin, Tian Jie, Metal–Organic Frameworks as a Theranostic Nanoplatform for Combinatorial Chemophotothermal Therapy Adapted to Different Administration, ACS Biomaterials Science & Engineering, 6, 2, 2020. Crossref

  33. Patil Mayuri B., Salve Priyanka M., Sonawane Shital V., Maru Avish D., Bhadane Jayshree S., Surawase Rajendra K., Technologies in Bilayer Tablet Manufacturing: A Review, Research Journal of Pharmaceutical Dosage Forms and Technology, 2021. Crossref

  34. Jauregizar Nerea, Quindós Guillermo, Gil-Alonso Sandra, Suárez Elena, Sevillano Elena, Eraso Elena, Postantifungal Effect of Antifungal Drugs against Candida: What Do We Know and How Can We Apply This Knowledge in the Clinical Setting?, Journal of Fungi, 8, 7, 2022. Crossref

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